Non-selective melanocortin receptor agonist (MC1R, MC3R, MC4R). MC4R activation drives sexual arousal and appetite suppression; MC1R drives melanogenesis.
Studies have administered: 0.25–1mg in research literature; titration from low doses noted in studies
Human studies demonstrate erection facilitation via MC4R in ED research. Significant skin tanning without UV exposure. Appetite suppression documented.
Nausea (common, especially initial doses), facial flushing, spontaneous erections, yawning, increased moles/nevi — carefully monitored in trials
These compounds have been examined together in research literature. Combination use is not endorsed or recommended — this information is provided for research context only.
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